关于 "Aryl Hydrocarbon Receptor" 的结果35+ 个结果
- GABAA receptor agent 1CAS: 1571-87-5
GABAA receptor agent 1 is a high affinity ligand for Gamma-aminobutyric acid A (GABAA) receptor that exerts potent anticonvulsant activity.
- Thrombin Receptor AntagonistCAS: 207553-92-2
The peptide T1, MSRPACPNDKYE, is based on the sequence of the thrombin receptor domain that functions as a tethered ligand for the receptor itself. T1 has been selected from a phage peptide library as an inhibitor of thrombin triggered platelet aggregation, serotonin release and tyrosine phosphorylation. Its anti-aggregatory activity was about ten-fold higher than that of the previously reported peptide antagonists of the thrombin receptor. MSRPACPNDKYE has served as model peptide in protein modification and MS studies.
- cFMS Receptor Inhibitor IVCAS: 959626-45-0
cFMS Receptor Inhibitor IV (Compound 42) 是一种有效的 cFMS 抑制剂，IC50 为 0.017 μM。
- A2B receptor antagonist 1CAS: 531506-36-2
A2Breceptorantagonist1是一个有效的A2B腺苷受体(A2Badenosinereceptor)拮抗剂，来自专利WO2009157938A1实例9B。
- S1p receptor agonist 1CAS: 1514888-56-2
S1p receptor agonist 1 是一种有效且具有口服活性的 S1P 受体激动剂，具有诱导 S1P1 内化的活性 (EC50=9.83 nM)。
- Androgen receptor antagonist 1CAS: 1338812-36-4
Androgenreceptorantagonist1是一种口服有效的完整雄激素受体(AR)拮抗剂，IC50为59nM。Androgenreceptorantagonist1可用于合成PROTACAR降解剂，1μM和10μMPROTACAR降解剂作用于LNCaP细胞，分别导致24%和47%AR蛋白降解。
| 货号 | 产品名称 | CAS号 | 靶点 / 通路 | 引用 | 结构 |
|---|---|---|---|---|---|
| GC60862 | GABAA receptor agent 1 | 1571-87-5 | GABA Receptor | ||
GABAA receptor agent 1 is a high affinity ligand for Gamma-aminobutyric acid A (GABAA) receptor that exerts potent anticonvulsant activity. | |||||
| GA23607 | Thrombin Receptor Antagonist | 207553-92-2 | - | ||
The peptide T1, MSRPACPNDKYE, is based on the sequence of the thrombin receptor domain that functions as a tethered ligand for the receptor itself. T1 has been selected from a phage peptide library as an inhibitor of thrombin triggered platelet aggregation, serotonin release and tyrosine phosphorylation. Its anti-aggregatory activity was about ten-fold higher than that of the previously reported peptide antagonists of the thrombin receptor.
MSRPACPNDKYE has served as model peptide in protein modification and MS studies. | |||||
| GC19170 | Glucagon receptor antagonists-4 | 1393124-08-7 | Glucagon Receptor | ||
A GCGR antagonist | |||||
| GC65976 | cFMS Receptor Inhibitor IV | 959626-45-0 | c-FMS | ||
cFMS Receptor Inhibitor IV (Compound 42) 是一种有效的 cFMS 抑制剂，IC50 为 0.017 μM。 | |||||
| GC19272 | Orexin 2 Receptor Agonist | 1796565-52-0 | OX Receptor | ||
An orexin 2 receptor agonist | |||||
| GC39554 | AT2 receptor agonist C21 | 477775-14-7 | Cardiomyopathy | ||
An AT2 receptor agonist | |||||
| GC31974 | A2B receptor antagonist 1 | 531506-36-2 | Adenosine Receptor | ||
A2Breceptorantagonist1是一个有效的A2B腺苷受体(A2Badenosinereceptor)拮抗剂，来自专利WO2009157938A1实例9B。 | |||||
| GC30759 | H3 receptor-MO-1 | 1240914-03-7 | Histamine Receptor | ||
H3receptor-MO-1是一种组胺H3受体(histamineH3receptor)调节剂。 | |||||
| GC31310 | H3 receptor antagonist 1 | 935840-13-4 | Histamine Receptor | ||
H3receptorantagonist1是组胺H3(histamineH3)受体拮抗剂，可用于神经疾病的研究。 | |||||
| GC19316 | S1p receptor agonist 1 | 1514888-56-2 | LPL Receptor | ||
S1p receptor agonist 1 是一种有效且具有口服活性的 S1P 受体激动剂，具有诱导 S1P1 内化的活性 (EC50=9.83 nM)。 | |||||
| GC60582 | Androgen receptor antagonist 1 | 1338812-36-4 | - | ||
Androgenreceptorantagonist1是一种口服有效的完整雄激素受体(AR)拮抗剂，IC50为59nM。Androgenreceptorantagonist1可用于合成PROTACAR降解剂，1μM和10μMPROTACAR降解剂作用于LNCaP细胞，分别导致24%和47%AR蛋白降解。 | |||||