关于 "Bromodomain" 的结果2 个结果

筛选:Signaling Pathways×
  • GC62654 structure
    GSK778
    CAS: 2451862-42-1

    GSK778 (iBET-BD1) is a strong BD1 bromodomain inhibitor of the BET proteins, with IC50 value of 75 nM for BRD2 BD1, 41 nM for BRD3 BD1, 41 nM for BRD4 BD1, and 143 nM for BRDT BD1.

  • GC25183 structure
    BZ1
    CAS: 2766623-38-3

    BZ1 (BPTF inhibitor, BPTF-IN-BZ1) is a pyridazinone-based BPTF (Bromodomain PHD Finger Transcription Factor) inhibitor with a high potency (Kd = 6.3 nM) and >350-fold selectivity over BET bromodomains.