关于 "Aurora Kinase" 的结果38+ 个结果
筛选:Signaling Pathways×
- Casein Kinase inhibitor A51CAS: 2079068-74-7
Casein Kinase inhibitor A51 是一种有效且具有口服活性的酪蛋白激酶 1α (CK1α) 抑制剂。Casein Kinase inhibitor A51 可诱导白血病细胞凋亡 (apoptosis),并具有有效的抗白血病活性。
- MAP kinase fragment [Multiple species]
Lys-Tyr-Ile-His-Ser-Ala-Asn-Val-Leu
- S6 Kinase Substrate Peptide 32
Measures the activity of kinases that phosphorylate ribosomal protein S6.
- Comprehensive Kinase Screening Library
For screening of a variety of kinase inhibitors
Signaling Pathways - PKCζ Pseudosubstrate InhibitorCAS: 799764-07-1
A substrate-competitive inhibitor of PKCζ activity
Signaling Pathways - Syk Inhibitor II (dihydrochloride)CAS: 227449-73-2
A selective blocker of spleen tyrosine kinase activity
Signaling Pathways - PKN3 Inhibitor Compound 16CAS: 2361545-75-5
PKN3 Inhibitor Compound 16是丝氨酸/苏氨酸蛋白激酶N3的抑制剂(IC50 = 14 nM)。
| 货号 | 产品名称 | CAS号 | 靶点 / 通路 | 引用 | 结构 |
|---|---|---|---|---|---|
| GC15711 | Aurora Kinase Inhibitor III | 879127-16-9 | Signaling Pathways | ||
A potent inhibitor of Aurora A kinase | |||||
| GC43624 | ERK Inhibitor | 1049738-54-6 | MAPK Signaling | ||
An ERK inhibitor | |||||
| GC45142 | VEGFR2 Kinase Inhibitor II | 288144-20-7 | Tyrosine Kinase | ||
A potent, cell-permeable inhibitor of VEGFR2 | |||||
| GC62442 | Casein Kinase inhibitor A51 | 2079068-74-7 | Apoptosis | ||
Casein Kinase inhibitor A51 是一种有效且具有口服活性的酪蛋白激酶 1α (CK1α) 抑制剂。Casein Kinase inhibitor A51 可诱导白血病细胞凋亡 (apoptosis),并具有有效的抗白血病活性。 | |||||
| GC49150 | Tpl2 Kinase Inhibitor (hydrochloride) | - | Innate Immunity | ||
A Tpl2 inhibitor | |||||
| GC71404 | hRIO2 kinase ligand-1 | 923841-73-0 | Others | ||
hRIO2 kinase ligand-1(com 9)是hRIO2激酶的配体,Kd值为520 nM。 | |||||
| GP10140 | MAP kinase fragment [Multiple species] | - | Cancer Biology Peptides | ||
Lys-Tyr-Ile-His-Ser-Ala-Asn-Val-Leu | |||||
| GP10104 | S6 Kinase Substrate Peptide 32 | - | S6 Kinase | ||
Measures the activity of kinases that phosphorylate ribosomal protein S6. | |||||
| GC44641 | PI3-Kinase α Inhibitor 2 | 371943-05-4 | PI3K/Akt/mTOR Signaling | ||
A PI3K p110α inhibitor | |||||
| GC46123 | Comprehensive Kinase Screening Library | - | Signaling Pathways | ||
For screening of a variety of kinase inhibitors | |||||
| GP10017 | [Ser25] Protein Kinase C (19-31) | 136795-05-6 | Neuroscience Peptides | ||
PKC substrate | |||||
| GC44642 | PI3-Kinase α Inhibitor 2 (hydrochloride) | 1188890-32-5 | PI3K/Akt/mTOR Signaling | ||
A PI3K p110α inhibitor | |||||
| GC43145 | Casein Kinase 2 Substrate (trifluoroacetate salt) | - | Signaling Pathways | ||
A peptide substrate for CK2 | |||||
| GC43128 | Calmodulin-Dependent Protein Kinase II (290-309) (trifluoroacetate salt) | - | Peptides | ||
A CaMKII inhibitor | |||||
| GC50253 | PF 543 hydrochloride | 1706522-79-3 | LPL Receptor | ||
A potent inhibitor of SPHK1 | |||||
| GC43676 | FLT3 Inhibitor III | 852045-46-6 | Tyrosine Kinase | ||
A potent, highly selective inhibitor of FLT3 | |||||
| GC43217 | CDK/CRK Inhibitor | 784211-09-2 | Signaling Pathways | ||
A CDK/CRK-specific kinase inhibitor | |||||
| GC43220 | Cdk5 Substrate | 164669-07-2 | Neuroscience | ||
A peptide substrate of Cdk5 | |||||
| GC52151 | PKCθ Inhibitor (hydrochloride) | 2253640-49-0 | Other Signal Transduction | ||
A PKCθ inhibitor | |||||
| GC44656 | PKCζ Pseudosubstrate Inhibitor | 799764-07-1 | Signaling Pathways | ||
A substrate-competitive inhibitor of PKCζ activity | |||||
| GC44979 | Syk Inhibitor II (dihydrochloride) | 227449-73-2 | Signaling Pathways | ||
A selective blocker of spleen tyrosine kinase activity | |||||
| GC91967 | LMTK3 Inhibitor C28 | 2764850-23-7 | Apoptosis | ||
LMTK3 Inhibitor C28是一种多激酶抑制剂。 | |||||
| GC49883 | DAPK Substrate Peptide (trifluoroacetate salt) | - | Apoptosis | ||
A DAPK1 peptide substrate | |||||
| GC92014 | PKN3 Inhibitor Compound 16 | 2361545-75-5 | Immunology/Inflammation | ||
PKN3 Inhibitor Compound 16是丝氨酸/苏氨酸蛋白激酶N3的抑制剂(IC50 = 14 nM)。 | |||||
