关于 "Virus Protease" 的结果41+ 个结果
- JNJ-67856633CAS: 2230273-76-2
JNJ-67856633 (JNJ-6633) is a potent, selective, allosteric inhibitor of MALT1 protease.
- Pepstatin Ammonium
Pepstatin Ammonium 是由放线菌类产生的一种特异性的天冬氨酸蛋白酶 (aspartic proteases) 抑制剂,能够抑制 hemoglobin-pepsin,hemoglobin-proctase,casein-pepsin,casein-proctase,casein-acid protease 和 hemoglobin-acid protease 的活性,IC50 值分别为 4.5 nM,6.2 nM,150 nM,290 nM,520 nM 和 260 nM;同时可抑制 HIV protease 的活性。
- AzvudineCAS: 1011529-10-4
Azvudine (RO-0622) is a novel nucleoside reverse transcriptase inhibitor with antiviral activity against human immunodeficiency virus (HIV), hepatitis B virus (HBV) and hepatitis C virus (HCV), potently inhibits HIV-1 (EC50 range 0.03 to 6.92 nM) and HIV-2 (EC50s ranging from 0.018 to 0.025 nM).
- Upamostat (WX-671)CAS: 590368-25-5
Upamostat (WX-671), a novel serine protease urokinase (uPA) inhibitor by inhibiting the urokinase-type plasminogen activator (uPA) system.
- Pepstatin Trifluoroacetate
Pepstatin Trifluoroacetate 是由放线菌类产生的一种特异性的天冬氨酸蛋白酶 (aspartic proteases) 抑制剂,能够抑制 hemoglobin-pepsin,hemoglobin-proctase,casein-pepsin,casein-proctase,casein-acid protease 和 hemoglobin-acid protease 的活性,IC50 值分别为 4.5 nM,6.2 nM,150 nM,290 nM,520 nM 和 260 nM。
| 货号 | 产品名称 | CAS号 | 靶点 / 通路 | 引用 | 结构 |
|---|---|---|---|---|---|
| GC37921 | Voxilaprevir | 1535212-07-7 | HCV Protease | ||
A pan-genotypic HCV NS3/4A protease inhibitor | |||||
| GC14454 | Tipranavir | 174484-41-4 | HIV | ||
A nonpeptidic HIV protease inhibitor | |||||
| GC13619 | JLK 6 | 62252-26-0 | Gamma Secretase | ||
A protease inhibitor | |||||
| GC62115 | JNJ-67856633 | 2230273-76-2 | MALT1 | ||
JNJ-67856633 (JNJ-6633) is a potent, selective, allosteric inhibitor of MALT1 protease. | |||||
| GC15785 | Saquinavir mesylate | 149845-06-7 | Autophagy | ||
An HIV protease inhibitor | |||||
| GC12945 | Atazanavir | 198904-31-3 | P-glycoprotein | ||
An inhibitor of HIV-1 protease | |||||
| GC14084 | Nelfinavir Mesylate | 159989-65-8 | HIV | ||
An HIV-1 protease inhibitor | |||||
| GC10959 | Boceprevir | 394730-60-0 | SARS-CoV | ||
An NS3/4A protease inhibitor | |||||
| GC36871 | Pepstatin Ammonium | - | Peptides | ||
Pepstatin Ammonium 是由放线菌类产生的一种特异性的天冬氨酸蛋白酶 (aspartic proteases) 抑制剂,能够抑制 hemoglobin-pepsin,hemoglobin-proctase,casein-pepsin,casein-proctase,casein-acid protease 和 hemoglobin-acid protease 的活性,IC50 值分别为 4.5 nM,6.2 nM,150 nM,290 nM,520 nM 和 260 nM;同时可抑制 HIV protease 的活性。 | |||||
| GC25117 | Azvudine | 1011529-10-4 | HCV Protease | ||
Azvudine (RO-0622) is a novel nucleoside reverse transcriptase inhibitor with antiviral activity against human immunodeficiency virus (HIV), hepatitis B virus (HBV) and hepatitis C virus (HCV), potently inhibits HIV-1 (EC50 range 0.03 to 6.92 nM) and HIV-2 (EC50s ranging from 0.018 to 0.025 nM). | |||||
| GC13716 | Lopinavir | 192725-17-0 | SARS-CoV | ||
A potent HIV-1 protease inhibitor | |||||
| GC17270 | Simeprevir | 923604-59-5 | HCV | ||
A potent NS3/4A protease inhibitor | |||||
| GC12299 | Telaprevir (VX-950) | 402957-28-2 | HCV | ||
An HCV NS3/4A protease inhibitor | |||||
| GC32882 | Upamostat (WX-671) | 590368-25-5 | Ser/Thr Protease | ||
Upamostat (WX-671), a novel serine protease urokinase (uPA) inhibitor by inhibiting the urokinase-type plasminogen activator (uPA) system. | |||||
| GC40256 | p-APMSF (hydrochloride) | 74938-88-8 | Proteolysis | ||
An irreversible inhibitor of serine proteases | |||||
| GC36872 | Pepstatin Trifluoroacetate | - | Peptides | ||
Pepstatin Trifluoroacetate 是由放线菌类产生的一种特异性的天冬氨酸蛋白酶 (aspartic proteases) 抑制剂,能够抑制 hemoglobin-pepsin,hemoglobin-proctase,casein-pepsin,casein-proctase,casein-acid protease 和 hemoglobin-acid protease 的活性,IC50 值分别为 4.5 nM,6.2 nM,150 nM,290 nM,520 nM 和 260 nM。 | |||||
| GC10155 | Vaniprevir | 923590-37-8 | HCV | ||
Vaniprevir (MK-7009) 是丙型肝炎病毒 (HCV) NS3/4A 蛋白酶的非共价竞争性抑制剂。 | |||||
