关于 "Nicotinic Receptor" 的结果31+ 个结果
- Nicotinic acid mononucleotide triethylamine
在 NAD+ 的生物合成中，Nicotinic acid mononucleotide triethylamine 通过烟酸磷酸核糖基转移酶由烟酸 (NA) 形成。Nicotinate mononucleotide triethylamine 是 nicotinamide mononucleotide/nicotinic acid mononucleotide 腺苷酰转移酶的底物。
Others - Nicotinic acid N-oxideCAS: 2398-81-4
Nicotinic acid N-oxide (Oxiniacic acid, Nicotinic acid 1-oxide) is nicotinic acid derivative that acts as a ligand and forms lead-carboxylate complexes having phosphorescent properties.
Others - Xanthinol NicotinateCAS: 437-74-1
Xanthinol Nicotinate (Complamin, Angioamin) is a potent vasodilator that can easily pass through the cell membrane and once inside the cell it causes an increase in glucose metabolism resulting in an increased energy.
Others - Methyl nicotinateCAS: 93-60-7
Methyl nicotinate (methyl pyridine-3-carboxylate) is an ester of methyl alcohol and nicotinic acid. It is a rubefacient.
Others - Myristyl nicotinateCAS: 273203-62-6
Myristyl nicotinate (Tetradecyl nicotinate) 是一种酯前药和 Nicotinic acid 的亲脂衍生物。Myristyl nicotinate 被开发用于将烟酸输送到皮肤中，以防止光化性角化病及其发展为皮肤癌。Myristyl nicotinate 显示刺激光损伤的皮肤中的表皮分化，增加皮肤 NAD 含量并增强人皮肤屏障。
Others - NOT Receptor Modulator 1CAS: 1015231-98-7
NOTReceptorModulator1是一种核受体NOT调节剂，详细信息请参考专利文献WO2008034974A1中Table1中的化合物Example39。
Others - Estrogen receptor modulator 1CAS: 63676-22-2
Estrogen receptor modulator 1 (compound 18) is an orally active and selective estrogen receptor modulator (SERM) with pIC50 of 0.46. Estrogen receptor modulator 1 exhibits potential anti-tumor activity.
- GPR34 receptor antagonist 2CAS: 907952-06-1
GPR34receptorantagonist2(CompoundD2)是GPR34受体拮抗剂，可用于免疫疾病，炎性疾病的研究。
Others - GPR52 receptor modulator 1CAS: 2642079-89-6
GPR52 receptor modulator 1(程序1)是一种GPR52受体调节剂，具有研究神经精神疾病的潜力。
Others - Succinate/succinate receptor antagonist 1CAS: 2361972-29-2
Succinate/succinate receptor antagonist 1 (compound 7a) 是一种琥珀酸受体拮抗剂。Succinate/succinate receptor antagonist 1 阻断牙龈组织中的琥珀酸信号。Succinate/succinate receptor antagonist 1 抑制琥珀酸受体 1 (SucnRl Antagonist 1) 的激活，IC50 值为 20 μμ。Succinate/succinate receptor antagonist 1 可用于牙周病的研究。
Others - Nanofin (2,6-Lupetidine)CAS: 504-03-0
Nanofin (2,6-Dimethylpiperidine, Lupetidine, Naniopinum) is a ganglion blocker alkaloid having nicotinic acetylcholine receptor antagonist action. It has antihypertensive effect used for mild to moderate hypertension.
Others
| 货号 | 产品名称 | CAS号 | 靶点 / 通路 | 引用 | 结构 |
|---|---|---|---|---|---|
| GC13206 | Nicotinic Acid | 59-67-6 | Endogenous Metabolite | ||
烟酸（维生素 B3）是一种具有口服活性的水溶性维生素 B3，是人体必需的营养素。 | |||||
| GC36739 | Nicotinic acid mononucleotide | 321-02-8 | Others | ||
A biosynthetic precursor to NAD | |||||
| GC69560 | Nicotinic acid mononucleotide triethylamine | - | Others | ||
在 NAD+ 的生物合成中，Nicotinic acid mononucleotide triethylamine 通过烟酸磷酸核糖基转移酶由烟酸 (NA) 形成。Nicotinate mononucleotide triethylamine 是 nicotinamide mononucleotide/nicotinic acid mononucleotide 腺苷酰转移酶的底物。 | |||||
| GC36740 | Nicotinic acid N-oxide | 2398-81-4 | Others | ||
Nicotinic acid N-oxide (Oxiniacic acid, Nicotinic acid 1-oxide) is nicotinic acid derivative that acts as a ligand and forms lead-carboxylate complexes having phosphorescent properties. | |||||
| GC39674 | Xanthinol Nicotinate | 437-74-1 | Others | ||
Xanthinol Nicotinate (Complamin, Angioamin) is a potent vasodilator that can easily pass through the cell membrane and once inside the cell it causes an increase in glucose metabolism resulting in an increased energy. | |||||
| GC36593 | Methyl nicotinate | 93-60-7 | Others | ||
Methyl nicotinate (methyl pyridine-3-carboxylate) is an ester of methyl alcohol and nicotinic acid. It is a rubefacient. | |||||
| GC12283 | Nicotine Difartrate | 65-31-6 | Others | ||
Nicotinic acetylcholine receptor (nAChR) agonist | |||||
| GC63815 | Benzyl nicotinate | 94-44-0 | Others | ||
Benzyl nicotinate 是一种血管扩张剂，用作引起充血的活性成分。 | |||||
| GC38822 | Myristyl nicotinate | 273203-62-6 | Others | ||
Myristyl nicotinate (Tetradecyl nicotinate) 是一种酯前药和 Nicotinic acid 的亲脂衍生物。Myristyl nicotinate 被开发用于将烟酸输送到皮肤中，以防止光化性角化病及其发展为皮肤癌。Myristyl nicotinate 显示刺激光损伤的皮肤中的表皮分化，增加皮肤 NAD 含量并增强人皮肤屏障。 | |||||
| GC40288 | (1'S,2'S)-Nicotine-1'-oxide | 51095-86-4 | Toxicology | ||
A nicotine metabolite | |||||
| GC67840 | Nicotinohydrazide | 553-53-7 | Others | ||
Nicotinohydrazide (Nicotinic acid hydrazide) 是一种小分子化合物。 | |||||
| GC16363 | TGR5 Receptor Agonist | 1197300-24-5 | GPCR19 | ||
A TGR5 agonist | |||||
| GC31192 | NOT Receptor Modulator 1 | 1015231-98-7 | Others | ||
NOTReceptorModulator1是一种核受体NOT调节剂，详细信息请参考专利文献WO2008034974A1中Table1中的化合物Example39。 | |||||
| GC60816 | Estrogen receptor modulator 1 | 63676-22-2 | Estrogen Receptor/ERR | ||
Estrogen receptor modulator 1 (compound 18) is an orally active and selective estrogen receptor modulator (SERM) with pIC50 of 0.46. Estrogen receptor modulator 1 exhibits potential anti-tumor activity. | |||||
| GC61596 | GPR34 receptor antagonist 2 | 907952-06-1 | Others | ||
GPR34receptorantagonist2(CompoundD2)是GPR34受体拮抗剂，可用于免疫疾病，炎性疾病的研究。 | |||||
| GC71309 | GPR52 receptor modulator 1 | 2642079-89-6 | Others | ||
GPR52 receptor modulator 1(程序1)是一种GPR52受体调节剂，具有研究神经精神疾病的潜力。 | |||||
| GC71325 | P2X7 receptor antagonist-4 | - | Others | ||
P2X7 receptor antagonist-4（化合物14a）是P2X7R拮抗剂。 | |||||
| GC71335 | GPR34 receptor antagonist 3 | - | Others | ||
GPR34 receptor antagonist 3（化合物5e）是一类GRP34拮抗剂，IC50为0.680μM。 | |||||
| GC90882 | ε-NAADP+ (sodium salt) | - | Nucleotides/Nucleosides | ||
一种荧光衍生物NAADP | |||||
| GC69966 | Succinate/succinate receptor antagonist 1 | 2361972-29-2 | Others | ||
Succinate/succinate receptor antagonist 1 (compound 7a) 是一种琥珀酸受体拮抗剂。Succinate/succinate receptor antagonist 1 阻断牙龈组织中的琥珀酸信号。Succinate/succinate receptor antagonist 1 抑制琥珀酸受体 1 (SucnRl Antagonist 1) 的激活，IC50 值为 20 μμ。Succinate/succinate receptor antagonist 1 可用于牙周病的研究。 | |||||
| GC45073 | TRAP-6 Peptide (trifluoroacetate salt) | - | Coagulation & Hemostasis | ||
A PAR1 agonist | |||||
| GC52436 | TRAP-6 amide (trifluoroacetate salt) | - | Immunology/Inflammation | ||
A peptide PAR1 agonist | |||||
| GC90543 | EGFR Peptide (human, mouse) (myristoylated) (trifluoroacetate salt) | - | MDR multidrug resistance | ||
一种PKC抑制剂 | |||||
| GC32508 | Nanofin (2,6-Lupetidine) | 504-03-0 | Others | ||
Nanofin (2,6-Dimethylpiperidine, Lupetidine, Naniopinum) is a ganglion blocker alkaloid having nicotinic acetylcholine receptor antagonist action. It has antihypertensive effect used for mild to moderate hypertension. | |||||