关于 "Nicotinic Receptor" 的结果24+ 个结果
- α-Conotoxin EICAS: 170663-33-9
Selective antagonist of neuromuscular nicotinic receptors α1β1γδ
Nicotinic Receptor - 5-Iodo-A-85380, 5-trimethylstannyl N-BOC derivativeCAS: 213766-21-3
Precursor to ligand for the α4β2 nicotinic receptor
Nicotinic Receptor - Sazetidine A dihydrochlorideCAS: 1197329-42-2
α4β2 nicotinic acetylcholine receptor ligand
Nicotinic Receptor - TMPH hydrochlorideCAS: 849461-91-2
neuronal nicotinic ACh receptors (nAChRs) antagonist
Nicotinic Receptor - 5-Iodo-A-85380 dihydrochlorideCAS: 1217837-17-6
α4β2 and α6β2 nicotinic acetylcholine receptors agonist
Nicotinic Receptor - (±)-Anatoxin A fumarateCAS: 1219922-30-1
(±)-Anatoxin A fumarate 是一种从淡水蓝藻中分离出来的天然生物碱。
Nicotinic Receptor - RJR-2403 oxalateCAS: 220662-95-3
RJR-2403 oxalate (RJR-2403 oxalate; (E)-Metanicotine oxalate) 是一种神经元烟碱受体激动剂,对 α4β2 亚型 (Ki=26 nM) 具有高选择性; > 1,000 倍的选择性比 α7 受体(Ki = 3.6 μM)。
- Mecamylamine hydrochlorideCAS: 826-39-1
Mecamylamine hydrochloride是一种非选择性、非竞争性的烟碱型乙酰胆碱受体(nAChR)拮抗剂,能够阻断多种不同的nAChR亚型,如α3β4、α4β2、α3β2,其IC 50 值分别为640nM、2.5μM、3.6μM。
- Varenicline HydrochlorideCAS: 230615-23-3
Varenicline Hydrochloride (CP 526555 hydrochloride) 是一种高亲和力、选择性的 α4β2 尼古丁乙酰胆碱受体 (nAChR) 部分激动剂和完整的 α7 nAChR 激动剂。
| 货号 | 产品名称 | CAS号 | 靶点 / 通路 | 引用 | 结构 |
|---|---|---|---|---|---|
| GC16302 | RuBi-Nicotine | 1256362-30-7 | Nicotinic Receptor | ||
Nicotinic receptor agonist | |||||
| GC15141 | ACV 1 | 740980-24-9 | Nicotinic Receptor | ||
Neuronal nicotinic receptor antagonist | |||||
| GC13644 | α-Conotoxin EI | 170663-33-9 | Nicotinic Receptor | ||
Selective antagonist of neuromuscular nicotinic receptors α1β1γδ | |||||
| GC14225 | 5-Iodo-A-85380, 5-trimethylstannyl N-BOC derivative | 213766-21-3 | Nicotinic Receptor | ||
Precursor to ligand for the α4β2 nicotinic receptor | |||||
| GC10575 | RJR-2403 hemioxalate | - | Nicotinic Receptor | ||
Neuronal nicotinic receptor agonist | |||||
| GC15132 | TC 1698 dihydrochloride | 700834-58-8 | Nicotinic Receptor | ||
nicotinic α7 receptor agonist | |||||
| GC14342 | Sazetidine A dihydrochloride | 1197329-42-2 | Nicotinic Receptor | ||
α4β2 nicotinic acetylcholine receptor ligand | |||||
| GC12237 | SIB 1508Y maleate | 192231-16-6 | Nicotinic Receptor | ||
neuronal nicotinic ACh receptor agonist | |||||
| GC11406 | TMPH hydrochloride | 849461-91-2 | Nicotinic Receptor | ||
neuronal nicotinic ACh receptors (nAChRs) antagonist | |||||
| GC11626 | 5-Iodo-A-85380 dihydrochloride | 1217837-17-6 | Nicotinic Receptor | ||
α4β2 and α6β2 nicotinic acetylcholine receptors agonist | |||||
| GC13052 | SR 16584 | 1150153-86-8 | Nicotinic Receptor | ||
Selective antagonist of α3β4 nicotinic acetylcholine receptors | |||||
| GC16927 | bPiDDB | 525596-66-1 | Nicotinic Receptor | ||
Orthosteric neuronal nicotinic acetylcholine receptor (nAChR) antagonist | |||||
| GC15383 | 4-Acetyl-1,1-dimethylpiperazinium iodide | 75667-84-4 | Nicotinic Receptor | ||
nicotinic agonist | |||||
| GC17060 | UB 165 fumarate | 200432-86-6 | Nicotinic Receptor | ||
Subtype-selective nicotinic agonist | |||||
| GC13366 | MG 624 | 77257-42-2 | Nicotinic Receptor | ||
An antagonist of neuronal nicotinic AChRs | |||||
| GC16937 | Carbamoylcholine chloride | 51-83-2 | nAChR | ||
Cholinergic receptor agonist | |||||
| GC17470 | (-)-Cotinine | 486-56-6 | Endogenous Metabolite | ||
A major metabolite of nicotine | |||||
| GC12774 | (±)-Anatoxin A fumarate | 1219922-30-1 | Nicotinic Receptor | ||
(±)-Anatoxin A fumarate 是一种从淡水蓝藻中分离出来的天然生物碱。 | |||||
| GC12102 | RJR-2403 oxalate | 220662-95-3 | nAChR | ||
RJR-2403 oxalate (RJR-2403 oxalate; (E)-Metanicotine oxalate) 是一种神经元烟碱受体激动剂,对 α4β2 亚型 (Ki=26 nM) 具有高选择性; > 1,000 倍的选择性比 α7 受体(Ki = 3.6 μM)。 | |||||
| GC14353 | α-Conotoxin ImI | 156467-85-5 | Nicotinic Receptor | ||
A conotoxin and an antagonist of α7 nAChRs | |||||
| GC18135 | Derquantel | 187865-22-1 | Nicotinic Receptor | ||
An anthelmintic spiroindole | |||||
| GC14157 | (-)-Lobeline hydrochloride | 134-63-4 | nAChR | ||
An alkaloid with diverse biological activities | |||||
| GC10329 | Mecamylamine hydrochloride | 826-39-1 | nAChR | ||
Mecamylamine hydrochloride是一种非选择性、非竞争性的烟碱型乙酰胆碱受体(nAChR)拮抗剂,能够阻断多种不同的nAChR亚型,如α3β4、α4β2、α3β2,其IC50值分别为640nM、2.5µM、3.6µM。 | |||||
| GC16143 | Varenicline Hydrochloride | 230615-23-3 | nAChR | ||
Varenicline Hydrochloride (CP 526555 hydrochloride) 是一种高亲和力、选择性的 α4β2 尼古丁乙酰胆碱受体 (nAChR) 部分激动剂和完整的 α7 nAChR 激动剂。 | |||||
