关于 "Nicotinic Receptor" 的结果67+ 个结果

Histamine H4 receptor antagonist-1是一种组胺H4受体拮抗剂，提取自专利WO2010108059A1化合物60。

Y1receptorantagonist1是H-409/22的一个异构体，是神经肽(neuropeptideY1)受体拮抗剂。

AMPA receptor modulator-1是一种强效、口服活性和选择性AMPAR调节蛋白TARPγ-8阴性调节剂，pIC50为9.7，比GluA1/γ-2更具选择性（pIC50=5）。

AMPA receptor antagonist-3是一种AMPA受体拮抗剂，从专利US20070027143A1中提取。

5-HT2A receptor agonist-3Ki=2.5nM、对5-HT2A的选择性是结构相似的5-HT2C受体的124倍。

Y1 receptor antagonist 1 formic （h409 -22异构体formic）是Y1受体拮抗剂1的甲酸盐形式。

Dopamine D2 receptor agonist-2(化合物36)是一种有效的多巴胺D2受体偏向性激动配体，Ki值为11.2 nM。

An NK 2 receptor antagonist

An NK 2 receptor antagonist

A peptide agonist of PAR1

A peptide agonist of PAR4

nicotinic α7 receptor agonist

α4β2 nicotinic acetylcholine receptor ligand

neuronal nicotinic ACh receptor agonist

neuronal nicotinic ACh receptors (nAChRs) antagonist

α4β2 and α6β2 nicotinic acetylcholine receptors agonist

Selective antagonist of α3β4 nicotinic acetylcholine receptors

Orthosteric neuronal nicotinic acetylcholine receptor (nAChR) antagonist

nicotinic agonist

PNU-282987 S enantiomer free base is the S-enantiomer of PNU-282987 free base, which is an α7 nicotinic acetylcholine receptor (α7 nAChR) agonist.

Subtype-selective nicotinic agonist

Lobelin sulphate (Lobeline sulfate, Bantron) is an alkaloid that has actions similar to nicotine on nicotinic cholinergic receptors but is less potent. It has a variety of therapeutic uses including in respiratory disorders, peripheral vascular disorders, insomnia, and smoking cessation.

An antagonist of neuronal nicotinic AChRs

α-Conotoxin GI, a 13-residue peptide originally isolated from the venom of the fish-hunting cone snail Conus geographus, acts as a competitive antagonist for the muscle-type nicotinic acetylcholine receptor (nAChR) with excellent selectivity for α/δ receptor subunit binding over α/γ.