关于 "c-RET" 的结果4 个结果
筛选:Metabolism×
- Varespladib (LY315920)CAS: 172732-68-2
Varespladib (LY315920)是一种强效、选择性的group IIA, nonpancreatic secretory PLA2 (sPLA2)抑制剂，IC 50 值为9nM。
- hnps-PLA InhibitorCAS: 185298-58-2
Hnps-PLA Inhibitor is an inhibitor of human nonpancreatic secretory Phospholipase A (hnps-PLA)
- YUM70CAS: 423145-35-1
YUM70 is a potent inhibitor of glucose-regulated protein 78 (GRP78) inhibitor with an IC50 of 1.5 μM. YUM70 induces endoplasmic reticulum (ER) stress-mediated apoptosis in pancreatic cancer.Although YUM70 inhibits GRP78 enzymatic activity, it increases the expression of GRP78 by increasing the chaperone translation mechanism.
| 货号 | 产品名称 | CAS号 | 靶点 / 通路 | 引用 | 结构 |
|---|---|---|---|---|---|
| GC44943 | sPLA2 Inhibitor | 393569-31-8 | Transcription Factors | ||
An orally active inhibitor of sPLA2-IIA | |||||
| GC17203 | Varespladib (LY315920) | 172732-68-2 | Phospholipase | ||
Varespladib (LY315920)是一种强效、选择性的group IIA, nonpancreatic secretory PLA2 (sPLA2)抑制剂，IC50值为9nM。 | |||||
| GC19745 | hnps-PLA Inhibitor | 185298-58-2 | Phospholipase | ||
Hnps-PLA Inhibitor is an inhibitor of human nonpancreatic secretory Phospholipase A (hnps-PLA) | |||||
| GC62388 | YUM70 | 423145-35-1 | Apoptosis | ||
YUM70 is a potent inhibitor of glucose-regulated protein 78 (GRP78) inhibitor with an IC50 of 1.5 μM. YUM70 induces endoplasmic reticulum (ER) stress-mediated apoptosis in pancreatic cancer.Although YUM70 inhibits GRP78 enzymatic activity, it increases the expression of GRP78 by increasing the chaperone translation mechanism. | |||||