关于 "Sigma Receptor" 的结果7+ 个结果
筛选:Metabolism×
- Glucagon Receptor Antagonist Inactive ControlCAS: 362482-00-6
An inactive control for glucagon receptor antagonist I
- Human Vitamin D Receptor Reporter Assay System
A nuclear receptor cell-based reporter assay
- Siramesine hydrochlorideCAS: 224177-60-0
Siramesine hydrochloride是一种有效的sigma-2受体激动剂。Siramesine对sigma-2受体具有亚纳摩尔亲和力 (IC 50 =0.12nM),并且对sigma-2受体的选择性是sigma-1受体的140倍(IC 50 =17nM)。
| 货号 | 产品名称 | CAS号 | 靶点 / 通路 | 引用 | 结构 |
|---|---|---|---|---|---|
| GC43765 | Glucagon Receptor Antagonist I | 438618-32-7 | Carbohydrate Metabolism | ||
A competitive antagonist of GCGR | |||||
| GC43766 | Glucagon Receptor Antagonist Inactive Control | 362482-00-6 | Carbohydrate Metabolism | ||
An inactive control for glucagon receptor antagonist I | |||||
| GC52504 | Human Vitamin D Receptor Reporter Assay System | - | Vitamin D Receptor | ||
A nuclear receptor cell-based reporter assay | |||||
| GC19508 | BLU-782 | 2141955-96-4 | ALK | ||
BLU-782 是一种口服精准疗法,专门设计用于选择性靶向突变体 ALK2。 | |||||
| GC15222 | Siramesine hydrochloride | 224177-60-0 | Ferroptosis | ||
Siramesine hydrochloride是一种有效的sigma-2受体激动剂。Siramesine对sigma-2受体具有亚纳摩尔亲和力 (IC50=0.12nM),并且对sigma-2受体的选择性是sigma-1受体的140倍(IC50=17nM)。 | |||||
| GC44999 | Tauro-α-muricholic Acid (sodium salt) | 2260905-08-4 | FXR & LXR | ||
An FXR receptor antagonist | |||||
| GC13083 | Siramesine | 147817-50-3 | Ferroptosis | ||
A selective σ2 receptor agonist | |||||
