关于 "Glucose Transporters" 的结果49+ 个结果

WZB117是一种靶向葡萄糖转运蛋白1（GLUT1）的小分子抑制剂。

A glucose transporter inhibitor

An inhibitor of glucose transport

DRB18 is a pan-GLUT (glucose transporters) inhibitor that inhibits growth and proliferation in several different cancer types with IC50 high nM range.

An inhibitor of monoamine transporters and OCTs

An inhibitor of sodium-glucose cotransporters

glutamate transport blocker

Inhibitor of BCRP multidrug transporter

glycine transporter 1 (GlyT1) inhibitor

glial glycine transporter (GlyT1) inhibitor

GABA transporter GAT-1 inhibitor

excitatory amino acid transporter (EAAT) blocker

excitatory amino acid transporter (EAAT) blocker

An inhibitor of L-glutamate transport

Potent equilibrative nucleoside transporter (ENT) inhibitor

Mitiglinide Calcium (KAD-1229) is a blood glucose-lowering drugs, stimulating insulin secretion by closing the ATP-sensitive K+ channels in pancreatic beta-cells.

An analog of anandamide which inhibits anandamide transport

Potent and selective inhibitor of the glial glycine transporter GlyT1b; active in vivo

FA16 is a ferroptosis inducer and an inhibitor of the system xc- cystine/glutamate transporter.

NBI-98782是一种强效且选择性的vesicular monoamine transporter 2 (VMAT2)抑制剂，K i 值为3nM。

Emamectin Benzoate (EMB, MK-244) activates gamma-amino butyric acid (GABA) transporter. Emamectin Benzoate induces of reactive oxygen species (ROS)-mediated DNA damage and apoptosis.

WAY-213613 is a potent, selective nonsubstrate reuptake inhibitor of GLT-1/EAAT2 with IC50 of 85 nM for excitatory amino acid transporter subtype 2 (EAAT2).

Valbenazine tosylate (NBI-98854) is the tosylate salt of valbenazine, a vesicular monoamine transporter 2 (VMAT2) inhibitor with a Ki value of 150 nM while displaying no significant binding to VAMT1(Ki<10 μM).

H100是一种氯离子运输(Cl-transport)抑制剂，可以部分抑制氯离子载体NaK2Clcotransporter和Band3anionexchanger，但是对KClcotransporter无作用。