关于 "Aldehyde dehydrogenase" 的结果7+ 个结果
筛选:Isocitrate Dehydrogenase (IDH)×
| 货号 | 产品名称 | CAS号 | 靶点 / 通路 | 引用 | 结构 |
|---|---|---|---|---|---|
| GC50129 | TC-E 5008 | 50405-58-8 | Isocitrate Dehydrogenase (IDH) | ||
Selective mutant isocitrate dehydrogenase 1 (mIDH1) inhibitor; phenotypically lethal | |||||
| GC10531 | AGI-5198 | 1355326-35-0 | Isocitrate Dehydrogenase (IDH) | ||
A potent, selective inhibitor of IDH1 mutations | |||||
| GC14757 | AGI-6780 | 1432660-47-3 | Isocitrate Dehydrogenase (IDH) | ||
A potent, selective inhibitor of mutant IDH2 | |||||
| GC17809 | GSK864 | 1816331-66-4 | Isocitrate Dehydrogenase (IDH) | ||
GSK864是一种突变型isocitrate dehydrogenases 1 (mIDH1)抑制剂,对IDH1 R132H、IDH1 R132C及WT IDH1的EC50值分别为0.16μM、0.10μM和2.74μM。 | |||||
| GC13147 | AG-221 (Enasidenib) | 1446502-11-9 | Isocitrate Dehydrogenase (IDH) | ||
An inhibitor of mutant IDH2 | |||||
| GC19380 | Vorasidenib | 1644545-52-7 | Isocitrate Dehydrogenase (IDH) | ||
An inhibitor of mutant IDH1 and IDH2 | |||||
| GC19059 | BAY-1436032 | 1803274-65-8 | Isocitrate Dehydrogenase (IDH) | ||
An inhibitor of mutant IDH1 | |||||
