关于 "Bromodomain" 的结果2 个结果

筛选:Immunology/Inflammation×
  • GC60182 structure
    GSK046
    CAS: 2474876-09-8

    A BD2 bromodomain inhibitor

  • GC62654 structure
    GSK778
    CAS: 2451862-42-1

    GSK778 (iBET-BD1) is a strong BD1 bromodomain inhibitor of the BET proteins, with IC50 value of 75 nM for BRD2 BD1, 41 nM for BRD3 BD1, 41 nM for BRD4 BD1, and 143 nM for BRDT BD1.