关于 "Bromodomain" 的结果2 个结果
筛选:Immunology/Inflammation×
| 货号 | 产品名称 | CAS号 | 靶点 / 通路 | 引用 | 结构 |
|---|---|---|---|---|---|
| GC60182 | GSK046 | 2474876-09-8 | Bromodomain | ||
A BD2 bromodomain inhibitor | |||||
| GC62654 | GSK778 | 2451862-42-1 | Apoptosis | ||
GSK778 (iBET-BD1) is a strong BD1 bromodomain inhibitor of the BET proteins, with IC50 value of 75 nM for BRD2 BD1, 41 nM for BRD3 BD1, 41 nM for BRD4 BD1, and 143 nM for BRDT BD1. | |||||
