关于 "Aurora Kinase" 的结果18+ 个结果
筛选:Immunology/Inflammation×
- Casein Kinase inhibitor A51CAS: 2079068-74-7
Casein Kinase inhibitor A51 是一种有效且具有口服活性的酪蛋白激酶 1α (CK1α) 抑制剂。Casein Kinase inhibitor A51 可诱导白血病细胞凋亡 (apoptosis),并具有有效的抗白血病活性。
- Syk Inhibitor II (dihydrochloride)CAS: 227449-73-2
A selective blocker of spleen tyrosine kinase activity
- PKN3 Inhibitor Compound 16CAS: 2361545-75-5
PKN3 Inhibitor Compound 16是丝氨酸/苏氨酸蛋白激酶N3的抑制剂(IC50 = 14 nM)。
Immunology/Inflammation - TrkB Agonist Prodrug R13CAS: 1609067-49-3
TrkB Agonist Prodrug R13(R13)是原肌球蛋白相关激酶B(TrkB)激活剂7,8-二羟基黄酮的前药形式。
- LY 294002 hydrochlorideCAS: 934389-88-5
Prototypical PI 3-kinase inhibitor; also inhibits other kinases
| 货号 | 产品名称 | CAS号 | 靶点 / 通路 | 引用 | 结构 |
|---|---|---|---|---|---|
| GC62442 | Casein Kinase inhibitor A51 | 2079068-74-7 | Apoptosis | ||
Casein Kinase inhibitor A51 是一种有效且具有口服活性的酪蛋白激酶 1α (CK1α) 抑制剂。Casein Kinase inhibitor A51 可诱导白血病细胞凋亡 (apoptosis),并具有有效的抗白血病活性。 | |||||
| GC49150 | Tpl2 Kinase Inhibitor (hydrochloride) | - | Innate Immunity | ||
A Tpl2 inhibitor | |||||
| GC18602 | p38 MAPK Inhibitor IV | 1638-41-1 | Innate Immunity | ||
An inhibitor of p38 MAP kinases | |||||
| GC50253 | PF 543 hydrochloride | 1706522-79-3 | LPL Receptor | ||
A potent inhibitor of SPHK1 | |||||
| GC44979 | Syk Inhibitor II (dihydrochloride) | 227449-73-2 | Signaling Pathways | ||
A selective blocker of spleen tyrosine kinase activity | |||||
| GC91148 | JAK Inhibitor 31 | 2891469-99-9 | JAK | ||
一种JAK2抑制剂 | |||||
| GC91967 | LMTK3 Inhibitor C28 | 2764850-23-7 | Apoptosis | ||
LMTK3 Inhibitor C28是一种多激酶抑制剂。 | |||||
| GC41740 | (S)-p38 MAPK Inhibitor III | 581098-48-8 | Innate Immunity | ||
A cell-permeable p38 MAP kinase inhibitor | |||||
| GC49883 | DAPK Substrate Peptide (trifluoroacetate salt) | - | Apoptosis | ||
A DAPK1 peptide substrate | |||||
| GC92014 | PKN3 Inhibitor Compound 16 | 2361545-75-5 | Immunology/Inflammation | ||
PKN3 Inhibitor Compound 16是丝氨酸/苏氨酸蛋白激酶N3的抑制剂(IC50 = 14 nM)。 | |||||
| GC91977 | TrkB Agonist Prodrug R13 | 1609067-49-3 | Behavioral Neuroscience | ||
TrkB Agonist Prodrug R13(R13)是原肌球蛋白相关激酶B(TrkB)激活剂7,8-二羟基黄酮的前药形式。 | |||||
| GC43176 | CAY10575 | 916985-21-2 | Transcription Factors | ||
An IKKβ and Plk1 inhibitor | |||||
| GC44880 | SD 1029 | 118372-34-2 | Hepatitis | ||
A JAK2 inhibitor | |||||
| GC50009 | LY 294002 hydrochloride | 934389-88-5 | Autophagy | ||
Prototypical PI 3-kinase inhibitor; also inhibits other kinases | |||||
| GC48971 | AZD 1152 (hydrochloride) | 722543-50-2 | Aurora Kinase | ||
A prodrug for a potent Aurora B inhibitor | |||||
| GC49903 | MRT67307 (hydrochloride) | 2095432-39-4 | Innate Immunity | ||
A kinase inhibitor | |||||
| GC50045 | PD 166285 dihydrochloride | 212391-63-4 | Apoptosis | ||
A tyrosine kinase inhibitor | |||||
| GC52516 | Erbstatin | 100827-28-9 | DNA Damage/DNA Repair | ||
A tyrosine kinase inhibitor | |||||
