关于 "Histone Acetyltransferases" 的结果15 个结果
筛选:Histone Acetyltransferases×
- CBP/p300-IN-3CAS: 2299226-01-8
P300/CBP-IN-3, a p300/CBP 组蛋白乙酰转移酶 (histone acetyltransferase) 抑制剂，化合物 6，来源于专利 WO 2019049061 A1。
Histone Acetyltransferases - NiCur
NiCur is a small molecule which blocks CREB-binding protein (CBP) histone acetyltransferase (HAT) activity and downregulates p53 activation upon genotoxic stress and diminishs the recruitment of p53 as well as RNA Polymerase II and levels of acetylation on histone H3 on CDKN1A promoter.
Histone Acetyltransferases - Histone H3 Peptide Substrate (1-21)
Target substrate for several histone modifying enzymes
Histone Acetyltransferases - KAT8 Inhibitor 19CAS: 28532-21-0
KAT8 inhibitor 19 is an inhibitor of lysine acetyltransferase 8 (KAT8; IC50 = 12.1 µM).
Histone Acetyltransferases - Butyrolactone 3CAS: 778649-18-6
Butyrolactone 3是组蛋白乙酰转移酶GCN5的小分子抑制剂（IC 50 = 100μM）。
Histone Acetyltransferases
| 货号 | 产品名称 | CAS号 | 靶点 / 通路 | 引用 | 结构 |
|---|---|---|---|---|---|
| GC12009 | HAT Inhibitor II | 932749-62-7 | Histone Acetyltransferases | ||
An inhibitor of HAT p300 | |||||
| GC45094 | TTK21 | 709676-56-2 | Behavioral Neuroscience | ||
An activator of CBP/p300 histone acetyltransferase activity | |||||
| GC17284 | Anacardic acid | 16611-84-0 | Epigenetic Reader Domain | ||
A histone acetyltransferase inhibitor | |||||
| GC38469 | CBP/p300-IN-3 | 2299226-01-8 | Histone Acetyltransferases | ||
P300/CBP-IN-3, a p300/CBP 组蛋白乙酰转移酶 (histone acetyltransferase) 抑制剂，化合物 6，来源于专利 WO 2019049061 A1。 | |||||
| GC62248 | NiCur | - | Histone Acetyltransferases | ||
NiCur is a small molecule which blocks CREB-binding protein (CBP) histone acetyltransferase (HAT) activity and downregulates p53 activation upon genotoxic stress and diminishs the recruitment of p53 as well as RNA Polymerase II and levels of acetylation on histone H3 on CDKN1A promoter. | |||||
| GC43837 | Histone H3 Peptide Substrate (1-21) | - | Histone Acetyltransferases | ||
Target substrate for several histone modifying enzymes | |||||
| GC91622 | KAT8 Inhibitor 19 | 28532-21-0 | Histone Acetyltransferases | ||
KAT8 inhibitor 19 is an inhibitor of lysine acetyltransferase 8 (KAT8; IC50 = 12.1 µM). | |||||
| GC15731 | L002 | 321695-57-2 | STAT | ||
A p300 acetyltransferase inhibitor | |||||
| GC11972 | NU 9056 | 1450644-28-6 | Histone Acetyltransferases | ||
NU 9056（1，2-双（异噻唑-5-基）二硫烷）是一种有效且选择性的Tip60（KAT5） 组蛋白乙酰转移酶（HAT）抑制剂，IC50值为2μM，具有抗肿瘤活性。 | |||||
| GC10226 | Butyrolactone 3 | 778649-18-6 | Histone Acetyltransferases | ||
Butyrolactone 3是组蛋白乙酰转移酶GCN5的小分子抑制剂（IC50 = 100μM）。 | |||||
| GC19891 | CTB | 451491-47-7 | Histone Acetyltransferases | ||
CTB 是一种有效的 p300 组蛋白乙酰转移酶激活剂 。 | |||||
| GC14524 | CTPB | 586976-24-1 | Histone Acetyltransferases | ||
A selective activator of p300 HAT | |||||
| GC13474 | Garcinol | 78824-30-3 | Other Apoptosis | ||
Garcinol是组蛋白乙酰转移酶p300和PCAF的非特异性抑制剂，IC50分别为7μM和5μM。 | |||||
| GC62104 | WM-3835 | 2229025-70-9 | Apoptosis | ||
WM-3835 is a novel and high-specific small molecule Lysine Acetyltransferase 7 (KAT7, MYST2, HBO1) inhibitor, able to potently suppressed OS cell proliferation and migration, and leads to apoptosis activation. | |||||
| GC11430 | Remodelin | 1622921-15-6 | Histone Acetyltransferases | ||
Remodelin 是 N-乙酰转移酶 10 (NAT10) 的小分子抑制剂。 | |||||