关于 "Endocrinology and Hormones" 的结果5+ 个结果
筛选:Chromatin/Epigenetics×
- Cl-amidineCAS: 913723-61-2
Cl-amidine is an irreversible pan-peptidylarginine deiminase (PAD) inhibitor with IC50 values of 5.9 ± 0.3 μM, 0.8 ± 0.3 μM, 6.2 ± 1.0 μM for PAD4, PAD1 and PAD3, respectively. Cl-amidine induces apoptosis.
| 货号 | 产品名称 | CAS号 | 靶点 / 通路 | 引用 | 结构 |
|---|---|---|---|---|---|
| GC35706 | Cl-amidine | 913723-61-2 | PAD | ||
Cl-amidine is an irreversible pan-peptidylarginine deiminase (PAD) inhibitor with IC50 values of 5.9 ± 0.3 μM, 0.8 ± 0.3 μM, 6.2 ± 1.0 μM for PAD4, PAD1 and PAD3, respectively. Cl-amidine induces apoptosis. | |||||
| GC16124 | Ruxolitinib phosphate | 1092939-17-7 | Mitophagy | ||
A potent and selective JAK1/JAK2 inhibitor | |||||
| GC13237 | LMK 235 | 1418033-25-6 | HDAC | ||
A selective inhibitor of HDAC4 and HDAC5 | |||||
| GC11209 | Cerdulatinib (PRT062070) | 1198300-79-6 | Spleen Tyrosine Kinase (Syk) | ||
A dual inhibitor of Syk and JAKs | |||||
| GC45927 | DS-437 | 1674364-87-4 | Histone Methyltransferase | ||
A dual inhibitor of PRMT5 and PRMT7 | |||||
