关于 "Histone Acetyltransferases" 的结果123+ 个结果

A p300 acetyltransferase inhibitor

NU 9056（1，2-双（异噻唑-5-基）二硫烷）是一种有效且选择性的Tip60（KAT5） 组蛋白乙酰转移酶（HAT）抑制剂，IC 50 值为2μM，具有抗肿瘤活性。

An inhibitor of JMJD2 histone demethylases

An inhibitor of G9a histone methyltransferase

A potent, cost-effective histone deacetylase inhibitor

A histone demethylase inhibitor

A highly potent inhibitor of G9a histone methyltransferase

Trapoxin A is a cyclotetrapeptide histone deacetylase (HDAC) inhibitor.

Inhibitor of histone deacetylases

EPZ-6438 是一种有效且具有生物利用度的 EZH2 抑制剂，EZH2 是多梳抑制复合物 2 (PRC2) 的催化亚基，可催化组蛋白 H3 (H3K27) 的赖氨酸 27 甲基化，从而抑制含有人 PRC2 的活性抑制常数 K i 值为 2.5 nM 的野生型 EZH2。

Butyrolactone 3是组蛋白乙酰转移酶GCN5的小分子抑制剂（IC 50 = 100μM）。

A G9a histone methyltransferase inhibitor

A potent inhibitor of G9a histone methyltransferase

EZM0414 is a potent, selective, and orally bioavailable inhibitor of Histone-lysine N-methyltransferase SETD2.

CTB 是一种有效的 p300 组蛋白乙酰转移酶激活剂 。

Selective inhibitor of KDM2/7 histone demethylases

An inhibitor of G9a histone methyltransferase

A G9a and GLP histone methyltransferase inhibitor

A selective activator of p300 HAT

Garcinol是组蛋白乙酰转移酶p300和PCAF的非特异性抑制剂，IC 50 分别为7μM和5μM。

PFI-90 is a selective inhibitor of the histone demethylase KDM3B. PFI-90 induces apoptosis and cell differentiation resulting in delayed tumor progression in vivo.

AMI-1 is a potent and specific Histone Methyltransferase (HMT) inhibitor with IC50 of 3.0 μM and 8.8 μM for yeast Hmt1p and human PRMT1, respectively.

CP2 is a cyclic peptide that inhibits the JmjC histone demethylases KDM4 with IC50 values of 42 nM and 29 nM for KDM4A and KDM4C, respectively.

FT895是组蛋白脱乙酰酶11（Histone Deacetylase 11，HDAC11）的有效选择性抑制剂，IC 50 值为3nM。