AChR
AChR(乙酰胆碱受体)
AChR, also known as acetylcholine receptor, is an integral membrane protein that responds to the binding of acetylcholine.
AChR 相关产品(53)
- GC14624Galanthamine HBrCAS: 1953-04-4
An alkaloid with AChE inhibitory and nAChR potentiating activities
- GC14703Oxybutynin chlorideCAS: 1508-65-2纯度: >98.00%
An antagonist of muscarinic acetylcholine receptors
- GC16059Tarafenacin D-tartrateCAS: 1159101-48-0纯度: >99.50%
Tarafenacin D-tartrate (SVT-40776 D-tartrate) 是一种高度选择性的 M3 毒蕈碱受体拮抗剂 (Ki= 0.19 nM),选择性是 M2 受体的约 200 倍。
- GC11128(±)-Vesamicol hydrochlorideCAS: 120447-62-3纯度: >99.00%
(±)-Vesamicol hydrochloride ((±)-AH5183 hydrochloride) 是一种有效的囊泡乙酰胆碱转运抑制剂,Ki 为 2 nM。
- GC16573GalanthamineCAS: 357-70-0纯度: >99.00%
An alkaloid with AChE inhibitory and nAChR potentiating activities
- GC17885VU0364572 (trifluoroacetate salt)CAS: 1240514-89-9
A selective muscarinic M 1 receptor agonist
| 货号 | 产品名称 | CAS号 | 纯度 | 结构 |
|---|---|---|---|---|
| GC14624 | Galanthamine HBr | 1953-04-4 | - | |
An alkaloid with AChE inhibitory and nAChR potentiating activities | ||||
| GC14703 | Oxybutynin chloride | 1508-65-2 | >98.00% | |
An antagonist of muscarinic acetylcholine receptors | ||||
| GC15014 | A-867744 | 1000279-69-5 | >99.50% | |
A positive allosteric modulator of α7 nAChRs | ||||
| GC15029 | Glycopyrrolate | 596-51-0 | >99.00% | |
A muscarinic acetylcholine receptor antagonist | ||||
| GC15150 | Tropicamide | 1508-75-4 | >99.00% | |
A selective muscarinic M 4 antagonist | ||||
| GC15178 | Hexamethonium Bromide | 55-97-0 | >98.00% | |
A nondepolarizing neuromuscular blocking agent | ||||
| GC16056 | Neostigmine Bromide | 114-80-7 | >98.00% | |
溴化新斯的明是一种胆碱酯酶抑制剂,用于治疗重症肌无力。 | ||||
| GC16059 | Tarafenacin D-tartrate | 1159101-48-0 | >99.50% | |
Tarafenacin D-tartrate (SVT-40776 D-tartrate) 是一种高度选择性的 M3 毒蕈碱受体拮抗剂 (Ki= 0.19 nM),选择性是 M2 受体的约 200 倍。 | ||||
| GC16255 | Decamethonium Bromide | 541-22-0 | >98.00% | |
A depolarizing neuromuscular blocking agent | ||||
| GC16526 | Atropine | 51-55-8 | >99.50% / >98.50% / >98.00% | |
A non-selective muscarinic acetylcholine receptor antagonist | ||||
| GC16635 | Diphemanil Methylsulfate | 62-97-5 | >98.00% | |
An anticholinergic agent | ||||
| GC16819 | VU0152100 | 409351-28-6 | >98.00% | |
A muscarinic M 4 receptor positive allosteric modulator | ||||
| GC17229 | Paroxetine HCl | 78246-49-8 | >99.50% / >99.00% | |
A selective serotonin reuptake inhibitor | ||||
| GC17483 | Trospium chloride | 10405-02-4 | >99.00% | |
An antagonist of muscarinic receptors | ||||
| GC17825 | Methscopolamine | 155-41-9 | - | |
A muscarinic acetylcholine receptor antagonist | ||||
| GC17908 | Homatropine Methylbromide | 80-49-9 | >98.00% | |
An anticholinergic agent | ||||
| GC10267 | Rivastigmine | 123441-03-2 | >98.00% | |
A cholinesterase inhibitor | ||||
| GC11128 | (±)-Vesamicol hydrochloride | 120447-62-3 | >99.00% | |
(±)-Vesamicol hydrochloride ((±)-AH5183 hydrochloride) 是一种有效的囊泡乙酰胆碱转运抑制剂,Ki 为 2 nM。 | ||||
| GC12507 | ML352 | 1649450-12-3 | >98.00% | |
An inhibitor of the presynaptic choline transporter | ||||
| GC13314 | L-Acetylcarnitine (hydrochloride) | 5080-50-2 | >98.00% | |
A mitochondrial metabolite | ||||
| GC13445 | LY2119620 | 886047-22-9 | >99.50% | |
LY2119620是一种muscarinic M 2 /M 4 受体选择性正性变构调节剂。 | ||||
| GC16573 | Galanthamine | 357-70-0 | >99.00% | |
An alkaloid with AChE inhibitory and nAChR potentiating activities | ||||
| GC17627 | Nitenpyram | 150824-47-8 | >99.50% | |
An insecticide | ||||
| GC17885 | VU0364572 (trifluoroacetate salt) | 1240514-89-9 | - | |
A selective muscarinic M 1 receptor agonist | ||||
