Remacemide

目录号: GC73886纯度: 不显示同义词: FPL 12924; PR 934-423; FPL 13592
Remacemide(FPL 12924)是一种口服活性、非竞争性、低亲和力NMDA受体拮抗剂。

Remacemide
Cas No.: 128298-28-2
规格价格库存数量操作
5 mg¥1,485.00现货
1
10 mg¥2,385.00现货
1
25 mg¥4,770.00现货
1

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产品描述 Description

Remacemide (FPL 12924) is an orally active, non-competitive, low-affinity NMDA receptor antagonist. Remacemide shows neuroprotection activity in animal models of poxia and ischemic stroke. Remacemide is also an anticonvulsant, and can be used in Parkinson's disease and Huntington's disease research.

References:
[1]. Schachter SC, et al. Remacemide: current status and clinical applications. Expert Opin Investig Drugs. 2000 Apr;9(4):871-83.
[2]. Dyker AG, et al. Remacemide drochloride: a double-blind, placebo-controlled, safety and tolerability study in patients with acute ischemic stroke. Stroke. 1999 Sep;30(9):1796-801.
[3]. Greenamyre JT, et al. Antiparkinsonian effects of remacemide drochloride, a glutamate antagonist, in rodent and primate models of Parkinson's disease. Ann Neurol. 1994 Jun;35(6):655-61.
[4]. Kieburtz K, et al. A controlled trial of remacemide drochloride in Huntington's disease. Mov Disord. 1996 May;11(3):273-7.

产品文档 Product Documents

Purity:不显示

化学性质Chemical Properties

CAS 号
128298-28-2
同义词
FPL 12924; PR 934-423; FPL 13592
分子式
C17H20N2O
分子量
268.35 g/mol
溶解性
DMSO : 87.5 mg/mL (326.07 mM; Need ultrasonic)
保存条件
-20°C
General tips
请根据产品在不同溶剂中的溶解度选择合适的溶剂配制储备液;一旦配成溶液,请分装保存,避免反复冻融造成的产品失效。
储备液的保存方式和期限:-80°C 储存时,请在 6 个月内使用,-20°C 储存时,请在 1 个月内使用。
为了提高溶解度,请将管子加热至 37°C,然后在超声波浴中震荡一段时间。
Shipping Condition
评估样品解决方案:配备蓝冰进行发货。所有其他可用尺寸:配备 RT,或根据请求配备蓝冰。

计算工具摩尔浓度 / 稀释 / 分子量 / 单位换算 / 体内配方 / 溶解度

g/mol