GlpBio

(Rac)-Tivantinib

目录号: GC74162纯度: >95.00%同义词: (Rac)-ARQ 197; (Rac)-ARQ 198
(Rac)-Tivantinib是Tivantinib的异构体，可以作为实验对照。
(Rac)-Tivantinib
Cas No.: 1239986-50-5
规格价格库存数量操作
5 mg¥554.00现货
1
10 mg¥886.00现货
1
50 mg¥2,546.00现货
1
100 mg¥3,874.00现货
1
10mM (in 1mL DMSO)¥608.00现货
1
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文献被引

本产品暂无引用记录;以下为 GlpBio 产品在 Nature / Cell / Science 等顶刊的客户引用样例
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    Cell
    187(9):2288-2304 (2024)
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    31, 1291–1307 (2021)

产品描述 Description

(Rac)-Tivantinib is the isomer of Tivantinib , and can be used as an experimental control. Tivantinib is a highly selective c-Met tyrosine kinase inhibitor with a Ki of 355 nM.

References:
[1]. Bai YL, et al. Quantitative analysis of tivantinib in rat plasma using ultra performance liquid chromatograp with tandem mass spectrometry. J Pharm Biomed Anal. 2016 Jul 15;126:98-102.
[2]. Munshi N, et al. ARQ 197, a novel and selective inhibitor of the human c-Met receptor tyrosine kinase with antitumor activity. Mol Cancer Ther. 2010 Jun;9(6):1544-53.

产品文档 Product Documents

Purity:>95.00%

化学性质Chemical Properties

CAS 号
1239986-50-5
同义词
(Rac)-ARQ 197; (Rac)-ARQ 198
分子式
C23H19N3O2
分子量
369.42 g/mol
溶解性
DMSO : 100 mg/mL (270.69 mM; Need ultrasonic)
保存条件
-20°C
General tips
请根据产品在不同溶剂中的溶解度选择合适的溶剂配制储备液；一旦配成溶液，请分装保存，避免反复冻融造成的产品失效。
储备液的保存方式和期限：-80°C 储存时，请在 6 个月内使用，-20°C 储存时，请在 1 个月内使用。
为了提高溶解度，请将管子加热至 37°C，然后在超声波浴中震荡一段时间。
Shipping Condition
评估样品解决方案：配备蓝冰进行发货。所有其他可用尺寸：配备 RT，或根据请求配备蓝冰。

计算工具摩尔浓度 / 稀释 / 分子量 / 单位换算 / 体内配方 / 溶解度

g/mol