PYCR1-IN-1

目录号: GC72970纯度: >98.00%
PYCR1-IN-1(化合物4)是吡咯啉-5-羧酸还原酶1(PYCR1)抑制剂,IC50为8.8µM。

PYCR1-IN-1
Cas No.: 709-85-3
规格价格库存数量操作
5 mg¥2,655.00现货
1
10 mg¥4,320.00现货
1

文献被引

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产品描述 Description

PYCR1-IN-1 (compound 4) is a pyrroline-5-carboxylate reductase 1 (PYCR1) inhibitor with an IC50 of 8.8 µM. PYCR1-IN-1 has anticancer effects.

References:
[1]. Kirsty Milne, et al. A fragment-like approach to PYCR1 inhibition. Bioorg Med Chem Lett. 2019 Sep 15;29(18):2626-2631.

产品文档 Product Documents

Purity:>98.00%Appearance:A liquid

化学性质Chemical Properties

CAS 号
709-85-3
分子式
C11H12BrN
分子量
238.12 g/mol
溶解性
DMSO : 100 mg/mL (419.96 mM; Need ultrasonic)
保存条件
4°C, stored under nitrogen
General tips
请根据产品在不同溶剂中的溶解度选择合适的溶剂配制储备液;一旦配成溶液,请分装保存,避免反复冻融造成的产品失效。
储备液的保存方式和期限:-80°C 储存时,请在 6 个月内使用,-20°C 储存时,请在 1 个月内使用。
为了提高溶解度,请将管子加热至 37°C,然后在超声波浴中震荡一段时间。
Shipping Condition
评估样品解决方案:配备蓝冰进行发货。所有其他可用尺寸:配备 RT,或根据请求配备蓝冰。

计算工具摩尔浓度 / 稀释 / 分子量 / 单位换算 / 体内配方 / 溶解度

g/mol