GlpBio

GV-150013

目录号: GC70255纯度: 不显示
GV-150013是一种选择性CCK-B受体拮抗剂。
GV-150013
Cas No.: 167355-22-8
规格价格库存数量操作
1 mg¥3,519.00现货
1
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文献被引

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    183(7):1867-1883 (2020)
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产品描述 Description

GV-150013 is a selective CCK-B receptor antagonist. GV-150013 has sleep aid effect.

GV-150013 (0.5 - 60μg/kg, ip, Once) increase REM sleep and non-REM sleep in old rats model[1].

References:
[1]. Crespi F. Cholecystokinin-B (CCK-B) receptor antagonists improve "aged" sleep: a new class of sleep modulators Methods Find Exp Clin Pharmacol. 1999 Jan-Feb;21(1):31-8.
[2]. F.Crespi, et al. Influence of cholecystokinin-B (CCK-B) receptor antagonists on rat electroencephalography (EEG): A new class of sleep modulators Gaviraghi. Dept of Pharmacology GlaxoWellcome S.p.A., Medicine Research Centre, via A. Fleming, 4, 37135 Verona, Italy

产品文档 Product Documents

Purity:不显示

化学性质Chemical Properties

CAS 号
167355-22-8
分子式
C33H34N4O3
分子量
534.65 g/mol
General tips
请根据产品在不同溶剂中的溶解度选择合适的溶剂配制储备液；一旦配成溶液，请分装保存，避免反复冻融造成的产品失效。
储备液的保存方式和期限：-80°C 储存时，请在 6 个月内使用，-20°C 储存时，请在 1 个月内使用。
为了提高溶解度，请将管子加热至 37°C，然后在超声波浴中震荡一段时间。
Shipping Condition
评估样品解决方案：配备蓝冰进行发货。所有其他可用尺寸：配备 RT，或根据请求配备蓝冰。

计算工具摩尔浓度 / 稀释 / 分子量 / 单位换算 / 体内配方 / 溶解度

g/mol